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CL 316243 disodium
CAS No. 138908-40-4
CL 316243 disodium ( CL316243 disodium )
产品货号. M11615 CAS No. 138908-40-4
CL 316243 is a potent, highly selective, orally active β3-adrenoceptor agonist with EC50 of 3 nM.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥1596 | 有现货 |
|
| 10MG | ￥2689 | 有现货 |
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| 25MG | ￥4520 | 有现货 |
|
| 50MG | ￥6383 | 有现货 |
|
| 100MG | ￥9072 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称CL 316243 disodium
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述CL 316243 is a potent, highly selective, orally active β3-adrenoceptor agonist with EC50 of 3 nM.
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产品描述CL 316243 is a potent, highly selective, orally active β3-adrenoceptor agonist with EC50 of 3 nM; Displays >10000-fold selective over β1 and β2 receptors; Significantly increases brown adipose tissue thermogenesis and resting metabolic rate in mice, also increases the concentration of insulin receptors and decreases the levels of serum insulin and blood glucose during the glucose overloading test.Obesity Discontinued
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同义词CL316243 disodium
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通路Angiogenesis
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靶点Adrenergic Receptor
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受体Adrenergic Receptor
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研究领域Metabolic Disease
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适应症Obesity
化学信息
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CAS Number138908-40-4
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分子量465.80
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分子式C20H18ClNNa2O7
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纯度>98% (HPLC)
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溶解度——
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SMILESCC(CC1=CC2=C(C=C1)OC(O2)(C(=O)[O-])C(=O)[O-])NCC(C3=CC(=CC=C3)Cl)O.[Na+].[Na+]
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化学全称5-[(2R)-2-[[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino]propyl]-1,3-benzodioxole-2,2-dicarboxylic acid disodium salt
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Berlan M, et al. J Pharmacol Exp Ther. 1994 Mar;268(3):1444-51.
2. Himms-Hagen J, et al. Am J Physiol. 1994 Apr;266(4 Pt 2):R1371-82.
3. Yoshida T, et al. Life Sci. 1994;54(7):491-8.
2. Himms-Hagen J, et al. Am J Physiol. 1994 Apr;266(4 Pt 2):R1371-82.
3. Yoshida T, et al. Life Sci. 1994;54(7):491-8.
产品手册
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